TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 880nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 1.47E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 1.50E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 1.20E+4nMAssay Description:Effect of Phosphatidylserine on inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 1.86E+4nMAssay Description:Inhibition of [3H]-PDBU binding to Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataKi: 4.10E+4nMAssay Description:Displacement of [3H]-phorbol-12,13-dibutyrate from rat brain protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 1.60nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 2.30nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/gamma type(Rattus norvegicus (Rat))
Nova Pharmaceutical
Curated by ChEMBL
Nova Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 2.70nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 2.85nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 3.10nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 3.80nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 4.60nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 8.80nMAssay Description:Inhibition of Protein kinase C alphaMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha type(Rattus norvegicus (Rat))
Temple University
Curated by PDSP Ki Database
Temple University
Curated by PDSP Ki Database
Affinity DataIC50: 30nMAssay Description:Binding affinity of protein kinase C (PKC).More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 99nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 222nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of Protein kinase C beta 1More data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 980nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetProtein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by ChEMBL
Kyowa Hakko Kogyo
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Binding affinity towards 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair